Mediated Rapid Aromatization of Dihydrobenzo[a]carbazole with their Scope and Limitations

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Benzo[a]carbazoles are rarely found in natural product and has unique position in biological active agents.1 Especially hydroxyl and amide derivatives of benzo[a]carabzole act as human Tpo receptor and antitumor agents respectively.2 Besides, some benzo[a]carbazoles used as molecular platforms for luminescent, hole-transporting and host material in organic light emitting diode.3 In general, transition metals are widely used for the synthesis of benzo[a]carbazole.4 Indeed, Fischer-Borsche is a classical method used for the preparation of benzo[a]carbazole.5 This involves the condensation of phenylhydrazine with tetralone followed by aromatization. However, aromatization of dihydrobenzo[a]carabzole is the challenging task. Such kind of transformations is carried out by heating the substrate with Pd/C in high boiling point solvents.6 Other organic based reagents capable of affecting the aromatization process are limited to quinone-derived reagent such as chloranil and DDQ.7 These kind of synthetic approaches required high temperature, loading of stoichiometric amounts of catalyst, long reaction time and low yield. For biological point of view, transition metals should be carefully removed from the final product. Also in the field of materials science, transition metallic impurities might influence the physical properties of the targeted material. To the best of our knowledge, very few reports are documented for the aromatization of dihydrobenzo[a]carbazoles to date. Therefore, development of rapid, efficient and conventional method for aromatization of dihydrobenzo[a]carbazoles is exceedingly desirable.
Over the last few decades, copper promoted transformations received considerable attention in organic syntheses.8 Moreover, copper...

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